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Pediatric cancer database
General information | Literature | Expression | Regulation | Variant | Interaction

Basic Information

Gene ID

2908

Name

NR3C1

Synonymous

GCCR|GCR|GR|GRL;nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor);NR3C1;nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor)

Definition

glucocorticoid nuclear receptor variant 1|glucocorticoid receptor|nuclear receptor subfamily 3 group C member 1 variant DL-1|nuclear receptor subfamily 3 group C member 1 variant NS-1

Position

5q31.3

Gene Type

protein-coding

Gene Regulation:

Transcription Factors
Post Translational Modification From dbPTM
Methylation Profile From DiseaseMeth database

Transcription Factors   [Top]

Regulation From TransFac database

GR-alpha(h) + Trx1(h) <==> GR-alpha(h):Trx1(h) (binding)
GR-alpha(h) --> CGA(h) (DNA binding).
GR-alpha(h) --> LYS(c) (DNA binding; transregulation).
GR-alpha(h) --> TAT(r) (DNA binding; transregulation).
GR-alpha(h) --> IL6(h) (DNA binding; transregulation).
c-Fos(h) + GR-alpha(h) <==> c-Fos(h):GR-alpha(h) (binding).
GR-alpha(h) + c-Jun(h) <==> GR-alpha(h):c-Jun(h) (binding).
Hsp90(h) + GR-alpha(h) <==> Hsp90(h):GR-alpha(h) (binding).
FKBP59(h) + GR-alpha(h) <==> FKBP59(h):GR-alpha(h) (binding).
hsp56(h) + GR-alpha(h) <==> hsp56(h):GR-alpha(h) (binding).
POU2F1(ha) + GR-alpha(h) <==> POU2F1(ha):GR-alpha(h) (binding).
GR-beta(h) + GR-alpha(h) <==> GR-beta(h):GR-alpha(h) (binding).
GR-alpha(h) --> IGFBP1(h) (DNA binding; transactivation).
GR-alpha(h) + GR-alpha(h) <==> GR-alpha(h):GR-alpha(h) (binding).
GR-alpha(h) + AP-1(h) <==> GR-alpha(h):AP-1(h) (binding).
POU2F1a(m) + GR-alpha(h) <==> POU2F1a(m):GR-alpha(h) (binding).
G-beta-2(h) + GR-alpha(h) <==> G-beta-2(h):GR-alpha(h) (binding)
GR-alpha(h) + G-beta-1(h) <==> GR-alpha(h):G-beta-1(h) (binding)
RACK1(h) + GR-alpha(h) <==> RACK1(h):GR-alpha(h) (binding)
GR-alpha(h) --> GR-alpha(h) (translocation)
GR-alpha(h) + 14-3-3sigma(h) <==> GR-alpha(h):14-3-3sigma(h) (binding)
GR-alpha(h) + 14-3-3eta(m.s.) <==> GR-alpha(h):14-3-3eta(m.s.) (binding)
GR-alpha(h) + DAP3(h) <==> GR-alpha(h):DAP3(h) (binding)
NF-IL6-3(h) + GR-alpha(h) <==> NF-IL6-3(h):GR-alpha(h) (binding)
GR-alpha(h) --> GR-alpha(h) (translocation)
GR-alpha(h) --/ IGFBP1(h) (DNA binding; transrepression).
GR-alpha(h) --> protein remnants (degradation)
GR-alpha(h) --> Wap(r) (transactivation)
NR3C1(h) --> GR-alpha(h) (expression).
relaxin-2(h) --> GR-alpha(h) (increase of abundance)
GR-alpha(h) --> GR-alpha(h) (translocation)
GR-alpha(h) --> GR-alpha(h) (translocation)
estradiol --/ GR-alpha(h) (decrease of abundance)
GR-beta(h) --> IL6(h) (DNA binding; transregulation).
GR-beta(h) --> TAT(r) (DNA binding; transregulation).
GR-beta(h) --> LYS(c) (DNA binding; transregulation).
GR-beta(h) --> CGA(h) (DNA binding).
GR-beta(h) + c-Fos(h) <==> GR-beta(h):c-Fos(h) (binding).
GR-beta(h) + c-Jun(h) <==> GR-beta(h):c-Jun(h) (binding).
GR-beta(h) + GR-alpha(h) <==> GR-beta(h):GR-alpha(h) (binding).
GR-beta(h) + FKBP59(h) <==> GR-beta(h):FKBP59(h) (binding).
GR-beta(h) + Hsp90(h) <==> GR-beta(h):Hsp90(h) (binding).
GR-beta(h) + hsp56(h) <==> GR-beta(h):hsp56(h) (binding).
GR-beta(h) + POU2F1(ha) <==> GR-beta(h):POU2F1(ha) (binding).
GR-beta(h) + AP-1(h) <==> GR-beta(h):AP-1(h) (binding).
GR-beta(h) + POU2F1a(m) <==> GR-beta(h):POU2F1a(m) (binding).
GR-beta(h) --> NR3C1(h) (DNA binding).
NR3C1(h) --> GR-beta(h) (expression).
relaxin-2(h) --> GR-beta(h) (increase of abundance)
GR(h) + 14-3-3eta(h) <==> GR(h):14-3-3eta(h) (binding)
GR(h) + PKAc(m) <==> GR(h):PKAc(m) (binding)
GR(h) --/ BGLAP(h) (DNA binding; transrepression).
GR(h) --> Orm1(m) (DNA binding).
GR(h) --> B1AR(s) (DNA binding).
GR(h) --> CRH(h) (DNA binding).
GR(h) --> GST-Y A2(r) (DNA binding).
GR(h) --> Aldh3a1(r) (DNA binding).
GR(h) --> AFP(h) (DNA binding; transactivation).
GR(h) --> CYP2C9(h) (DNA binding; transactivation).
GR(h) + STAT5A(m) <==> GR(h):STAT5A(m) (binding)
GR(h) --> NR1I3(h) (DNA binding).
GR(h) + MVP(h) <==> GR(h):MVP(h) (binding)
GR(h) + DP97-xbb2(h) <==> GR(h):DP97-xbb2(h) (binding)
PIAS2(m.s.) + GR(h) <==> PIAS2(m.s.):GR(h) (binding)
ELL(m.s.) + GR(h) <==> ELL(m.s.):GR(h) (binding)
ASC-2(r) + GR(h) <==> ASC-2(r):GR(h) (binding)
ASC-2(h) + GR(h) <==> ASC-2(h):GR(h) (binding)
GT198(r) + GR(h) <==> GT198(r):GR(h) (binding)
GR(h) + GT198(h) <==> GR(h):GT198(h) (binding)
GR(h) + relaxin(h) <==> GR(h):relaxin(h) (binding)
Hsp70(h) + GR(h) <==> Hsp70(h):GR(h) (binding)
Hsp90(h) + GR(h) <==> Hsp90(h):GR(h) (binding)
GR(h) + RIP140(h) <==> GR(h):RIP140(h) (binding)
14-3-3eta(h) + GR(h) <==> 14-3-3eta(h):GR(h) (binding)
RIP140(h) + GR(h) + 14-3-3eta(h) <==> RIP140(h):GR(h):14-3-3eta(h) (binding)
GR(h) + DRIP205-isoform4(m) <==> GR(h):DRIP205-isoform4(m) (binding)
GR(h) + SRC3(h) <==> GR(h):SRC3(h) (binding)
GR(h) + SRC-1(h) <==> GR(h):SRC-1(h) (binding)
GR(h) + TIF2(m) <==> GR(h):TIF2(m) (binding)
GR(h) + RXR-alpha(h) <==> GR(h):RXR-alpha(h) (binding)
GR(h) + G-beta(h) <==> GR(h):G-beta(h) (binding)
GR(h) + G-gamma(h) <==> GR(h):G-gamma(h) (binding)
SRP1alpha(m) + GR(h) <==> SRP1alpha(m):GR(h) (binding)
importin-7(x) + GR(h) <==> importin-7(x):GR(h) (binding)
GR(h) + importin-8(h) <==> GR(h):importin-8(h) (binding)
GR(h) --> UGT1A1(h) (DNA binding).
GR(h) --> GR(h) (translocation)
NF-kappaB1-isoform1(h) + GR(h) <==> NF-kappaB1-isoform1(h):GR(h) (binding)
RelA-p65(h) + GR(h) <==> RelA-p65(h):GR(h) (binding)
TRAP170(m.s.) + GR(h) <==> TRAP170(m.s.):GR(h) (binding)
DRIP205(m.s.) + GR(h) <==> DRIP205(m.s.):GR(h) (binding)
GR(h) --> Pnmt(r) (DNA binding; transactivation).
GR(h) --> NR3C1(h) (DNA binding).
GR(h) + hnRNPA1(h) <==> GR(h):hnRNPA1(h) (binding)
GR(h) --> CSH1(h) (DNA binding).
GR(h) --> CD38(h) (DNA binding).
ska2(h) + GR(h) <==> ska2(h):GR(h) (binding)
GR(h) + ska2(m.s.) <==> GR(h):ska2(m.s.) (binding)
GR(h) --/ POMC(h) (transrepression)
GR(h) --> Orm2(m) (DNA binding; transactivation).
GR(h) --> PLA2G4A(h) (DNA binding).
GR(h) + HNF-4alpha(h) <==> HNF-4alpha(h):GR(h) (binding)
GR(h) --> Agtr1b(r) (DNA binding).
GR(h) --> FKBP5(h) (DNA binding).
NR3C1(h) --> GR(h) (expression).
ARA70(m.s.) --> GR(h) (activation)
PIAS2(m.s.) --> GR(h) (regulation of protein activity)
GR(h) --> GR(h) (translocation)
NR3C1(h) --> GR-Alpha-2(h) (expression).
NR3C1(h) --> GR-Beta-2(h) (expression).
NR3C1(h) --> GR-Abeta(h) (expression).

Post Translational Modification   [Top]

Location (AA)

PTM type

Literature

Database

113Phosphoserine (By similarity).Swiss-Prot 53.0
141Phosphoserine (By similarity).Swiss-Prot 53.0
203Phosphoserine.Swiss-Prot 53.0
211Phosphoserine.Swiss-Prot 53.0
226Phosphoserine (By similarity).Swiss-Prot 53.0
277Glycyl lysine isopeptide (Lys-Gly)(interchain with G-Cter in SUMO).Swiss-Prot 53.0
293Glycyl lysine isopeptide (Lys-Gly)(interchain with G-Cter in SUMO).Swiss-Prot 53.0
508Phosphoserine (DNA-PK)9038175Phospho.ELM 6.0
203Phosphoserine12000743Phospho.ELM 6.0
211Phosphoserine15817653Phospho.ELM 6.0
141Phosphoserine7873448;2019585Phospho.ELM 6.0
113Phosphoserine7873448;2019585Phospho.ELM 6.0

Methylation Profile   [Top]

Chromosome

Location

Source

chr5

Promoter: 142763738 - 142765738Agilent_014791

chr5

Promoter: 142762947 - 142764947Agilent_014791

chr5

Promoter: 142762947 - 142764947GSE27584

chr5

Promoter: 142763738 - 142765738GSE27584

chr5

Promoter: 142762947 - 142764947GSE27584

chr5

Promoter: 142762947 - 142764947GSE27584

chr5

Promoter: 142762947 - 142764947Agilent_014791_44K

chr5

Promoter: 142762947 - 142764947PMID:17167179

chr5

Promoter: 142794770 - 142796770PMID:17167179

chr5

Promoter: 142794770 - 142796770PMID:17167179

chr5

Promoter: 142763738 - 142765738PMID:17167179

chr5

Promoter: 142794770 - 142796770PMID:17167179

chr5

Promoter: 142762947 - 142764947PMID:17167179

chr5

Promoter: 142762947 - 142764947PMID:17167179


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