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Cell senescence database
General information | Literature | Expression | Regulation | Mutation | Homolog | Interaction

Basic Information

Gene ID

5604

Name

MAP2K1

Synonymous

mitogen-activated protein kinase kinase 1;MAP2K1;mitogen-activated protein kinase kinase 1

Definition

ERK activator kinase 1|MAPK/ERK kinase 1|MAPKK 1|MEK 1|dual specificity mitogen-activated protein kinase kinase 1|protein kinase, mitogen-activated, kinase 1 (MAP kinase kinase 1)

Position

15q22.1-q22.33

Gene Type

protein-coding

Gene Regulation:

Transcription Factors
Post Transcriptional Modification From dbPTM
Methylation Profile From DiseaseMeth database

Transcription Factors   [Top]

Regulation From TransFac database

MEK1(h) + ATP --H-Ras(h):GTP:NO:Raf-1(h)--> MEK1(h){p} + ADP (phosphorylation)
Raf-1(h) + MEK1(h) <==> Raf-1(h):MEK1(h) (binding)
MEK1(h) + ATP --> MEK1(h){p} + ADP (phosphorylation)
MEK1(h) + ATP --Lck(m.s.)--> MEK1(h){pY} + ADP (phosphorylation)
MEK1(h) + Raf-1(h) <==> MEK1(h):Raf-1(h) (binding)
Grb10zeta(h) + MEK1(h) <==> Grb10zeta(h):MEK1(h) (binding)
MEK1(h) --> E47(h){p} (increase of phosphorylation)
MEK1(h) --> E47(m){p} (increase of phosphorylation)
MEK1(h) --/ E47(h) (decrease of abundance)
MEK1(h) --> E47(h){p}:Skp2(h) (increase of binding)
MEK1(h) --> BIRC3(h) (transactivation)
MEK1(h) --> MICA(h) (increase of abundance)
MEK1(h) + PPARgamma(h) <==> MEK1(h):PPARgamma(h) (binding)
MEK1(h) + ATP --> MEK1(h){pS} + ADP (phosphorylation)
MEK1(h) --/ NOTCH1(h) (transrepression)
MAP2K1(h) --> MEK1(h) (expression).
CSE1(h) + ATP --MEK1(h)--> CSE1(h){pY} + ADP (phosphorylation)
ERK1(m) + ATP --MEK1(h)--> ERK1(m){p} + ADP (phosphorylation)
ERK2(m) + ATP --MEK1(h)--> ERK2(m){p} + ADP (phosphorylation)
ERK1(h) + ATP --MEK1(h)--> ERK1(h){p} + ADP (phosphorylation)
ERK2(h) + ATP --MEK1(h)--> ERK2(h){p} + ADP (phosphorylation)
MEK1(h) + 2 ATP --> MEK1(h){pS218}{pS222} + 2 ADP (phosphorylation)
MEK1(h) + ATP --Cot(h){p}--> MEK1(h){p} + ADP (phosphorylation)
MEK1(h) + PPARgamma1(m.s.) <==> MEK1(h):PPARgamma1(m.s.) (binding)
MEK1(h) + PPARgamma1(h) <==> MEK1(h):PPARgamma1(h) (binding)
MEK1(h) + PPARgamma(m.s.) <==> MEK1(h):PPARgamma(m.s.) (binding)
MEK1(h) + ATP --Cdk5(h)--> MEK1(h){p} + ADP (phosphorylation)
ERK2(r) + MEK1(h) <==> ERK2(r):MEK1(h) (binding)
ERK1(h) + MEK1(h) <==> ERK1(h):MEK1(h) (binding)
ERK2(r) + MEK1(h) <==> ERK2(r):MEK1(h) (binding)
MAP2K1(h) --> MEK1(h) (expression).
HCV-NS5A(HCV) + ATP --MEK1(h)--> HCV-NS5A(HCV){p} + ADP (phosphorylation)
ERK2(r) + ATP --MEK1(h)--> ERK2(r){p} + ADP (phosphorylation)

Post Transcriptional Modification   [Top]

Location (AA)

PTM type

Literature

Database

218Phosphoserine (by RAF).Swiss-Prot 53.0
222Phosphoserine (by RAF).Swiss-Prot 53.0
221Phosphoserine (MAP3K8;MAP3K)94178255;15175348;7624324;8039496;15466476;8131746Phospho.ELM 6.0
217Phosphoserine (MAP3K8;MAP2K)94178255;7873542;7936666;7624324;15466476;8131746Phospho.ELM 6.0
385Phosphothreonine (MAPK1)10567369Phospho.ELM 6.0
211Phosphoserine12506122Phospho.ELM 6.0
291Phosphothreonine (MAPK1)10567369;9351825Phospho.ELM 6.0

Methylation Profile   [Top]

Chromosome

Location

Source

chr15

Promoter: 64465179 - 64467179Agilent_014791

chr15

Promoter: 64465179 - 64467179GSE27584

chr15

Promoter: 64465179 - 64467179Agilent_014791_44K


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