Pediatric cancer gene database (Pedican) Home
Pedican
Pediatric cancer database
General information | Literature | Expression | Regulation | Variant | Interaction

Basic Information

Gene ID

2149

Name

F2R

Synonymous

CF2R|HTR|PAR-1|PAR1|TR;coagulation factor II (thrombin) receptor;F2R;coagulation factor II (thrombin) receptor

Definition

coagulation factor II receptor|protease-activated receptor 1|proteinase-activated receptor 1|thrombin receptor

Position

5q13

Gene Type

protein-coding

Gene Regulation:

Transcription Factors
Post Translational Modification From dbPTM
Methylation Profile From DiseaseMeth database

Transcription Factors   [Top]

Regulation From TransFac database

PAR-1(h) --> Gi(v.s.) (activation)
PAR-1(h) --> Gq(v.s.) (activation)
PAR-1(h) --> Vav(h){pY} (increase of phosphorylation)
PAR-1(h) --> ZAP-70(h){pY} (increase of phosphorylation)
PAR-1(h) --> SLP-76(h){pY} (increase of phosphorylation)
PAR-1(h) --> IL8(h) (transactivation)
PAR-1(h) --> IKK(h){p} (increase of phosphorylation)
PAR-1(h) --> cytosolic phospholipase A2(h){p} (increase of phosphorylation)
PAR-1(h) --> FAK1(h){pY} (increase of phosphorylation)
PAR-1(h) --> arachidonic acid (increase of secretion)
PAR-1(h) --> ERK2(h){p} (increase of phosphorylation)
F2R(h) --> PAR-1(h) (expression).
F2R(h) --> PAR-1(h) (expression).

Post Translational Modification   [Top]

Location (AA)

PTM type

Literature

Database

35N-linked (GlcNAc...) (Potential).Swiss-Prot 53.0
62N-linked (GlcNAc...) (Potential).Swiss-Prot 53.0
75N-linked (GlcNAc...) (Potential).Swiss-Prot 53.0
250N-linked (GlcNAc...) (Potential).Swiss-Prot 53.0
259N-linked (GlcNAc...) (Potential).Swiss-Prot 53.0
410Phosphothreonine8955127Phospho.ELM 6.0
425Phosphothreonine8955127Phospho.ELM 6.0
375Phosphoserine8955127Phospho.ELM 6.0
376Phosphoserine8955127Phospho.ELM 6.0
384Phosphoserine8955127Phospho.ELM 6.0
391Phosphoserine8955127Phospho.ELM 6.0
392Phosphoserine8955127Phospho.ELM 6.0
395Phosphoserine8955127Phospho.ELM 6.0
396Phosphoserine8955127Phospho.ELM 6.0
399Phosphoserine8955127Phospho.ELM 6.0
400Phosphoserine8955127Phospho.ELM 6.0
406Phosphoserine8955127Phospho.ELM 6.0
413Phosphoserine8955127Phospho.ELM 6.0
412Phosphoserine8955127Phospho.ELM 6.0
418Phosphoserine8955127Phospho.ELM 6.0
397Phosphotyrosine8955127Phospho.ELM 6.0
383Phosphotyrosine15023990Phospho.ELM 6.0

Methylation Profile   [Top]

Chromosome

Location

Source

chr5

Promoter: 76046047 - 76048047Agilent_014791

chr5

Promoter: 76046047 - 76048047GoldenGate_Methylation_Cancer_Panel_I

chr5

Promoter: 76046047 - 76048047GSE27584

chr5

Promoter: 76046047 - 76048047Agilent_014791_44K

chr5

Promoter: 76046047 - 76048047PMID:16367923


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